最近の発表論文(2011年8月18日更新)
- Direct
ethoxycarbonyldifluoromethylation of aromatic compounds
using Fenton reagent; Y. Ohtsuka, T. Yamakawa, Tetrahedron,
Vol.67,
No.12, p2323-2331 (2011).
- 遷移金属触媒を用いた芳香族化合物への含フッ素官能基導入法; 井上宗宣, 荒木啓介, 月刊ファインケミカル, Vol.40, No.1, p40-45
(2011).
- 発展を続けるフッ素化学−総論; 井上宗宣, 月刊ファインケミカル, Vol.40, No.1, p5-6
(2011).
- クロスカップリングによる含フッ素官能基導入反応; 井上宗宣, 荒木啓介, クロスカップリング反応−基礎と産業応用−第16章, p210-216 (2010).
- Synthesis and
Electroluminescence of New Organic Emitters Based on a π-Conjugated 1,3,5-Triazine
Core; H. Aihara, T. Tanaka, M. Sato and T. Yamakawa, Transactions
of the Materials Research Society of Japan, Vol.35,
No.3, p675-680 (2010).
- 化学的にみた抗うつ薬とその薬理; 諸岡良彦, 平井憲次, 渡部勇信, 臨床精神薬理, Vol.13, No.6, p1223-1237
(2010).
- Diverse dimerization
of molecular tweezers with a
2,4,6-triphenyl-1,3,5-triazine spacer in the solid state;
Y. Hisamatsu and H. Aihara, Chemical Communication,
Vol.46, No.27, p4902-4904 (2010).
- Convenient screening
of 4-hydroxyphenylpyruvate dioxygenase inhibitors by UV
absorbance detection in the presence of Fe2+
ion; Y. Ikeda, R. Ohno and Y. Sato, Journal of
Pesticide Science, Vol.35, No.3, p321-325 (2010).
- A novel synthesis of
the 2-amino-1H-imidazol-4-carbaldehyde derivatives and
its application to the efficient synthesis of
2-aminoimidazole alkaloids, oroidin, hymenidin,
dispacamide, monobromodispacamide, and ageladine A; N. Ando and S. Terashima, Tetrahedron,
Vol.66,
No.32, p6224-6237 (2010).
-
- Synthesis and insecticidal activity of novel
1-alkyl-3-sulfonyloxypyrazole- 4-carboxamide derivatives;
R. Ohno, M. Nagaoka, K. Hirai, A. Uchida, S. Kochi, O.
Yamada, J. Tokumura, Journal of Pesticide Science,
Vol.35, No.1, p15-22 (2010).
- High electron mobility layers of triazines for improving
driving voltages, power conversion efficiencies, and
operational stability of organic light-emitting diodes:
T. Matsushima, M. Takamori, Y. Miyashita, Y. Honma, T.
Tanaka, H. Aihara and H. Murata, Organic Electronics,
Vol.11, No.1, p16-22 (2010).
- Possible Biosynthetic Pathways for all cis-3,6,9,12,15,19,22,25,28-Hentriacontanonaene
in Bacteria; S. Sugihara, R. Hori, H. Nakanowatari, Y.
Takada, I. Yumoto, N. Morita, Y. Yano, K. Watanabe and H.
Okuyama, Lipids, Vol.45, No.2, p167-177 (2010).
- Trifluoromethylation of various aromatic compounds by CF3I
in the presence of Fe(U) compound, H2O2
and dimethylsulfoxide; T. Kino, Y. Nagase, Y. Ohtsuka, K.
Yamamoto, D. Uraguchi, K. Tokuhisa, T. Yamakawa, Journal
of Fluorine Chemistry, Vol.131, No.1, p98-105 (2010).
- 触媒的含フッ素アルキル基およびアルケニル基の有機化合物への導入;
山川哲, ファインケミカル, Vol.39, No.1,
p22-26(2010).
- A New Quadruple Hydrogen-Bonding Module with a DDAA
Array: Formation of a Stable Homodimer without
Competition from Undesired Hydrogen-Bonded Dimers; Y.
Hisamatsu, N. Shirai, S. Ikeda and K. Odashima, Organic
Letters, Vo.11, No.19, p4342?4345 (2009).
- pfaB products determine the molecular species
produced in bacterial polyunsaturated fatty acid
biosynthesis; Y. Orikasa, M. Tanaka, S. Sugihara, R.
Hori, T. Nishida*, A. Ueno, N. Morita, Y. Yano, K.
Yamamoto, A. Shibahara, H. Hayashi, Y. Yamada, A. Yamada,
R. Yu, K. Watanabe & H. Okuyama, FEMS Microbiology
Letters, Vol.295, No.2, p170-176 (2009).
- 仮想スクリーニング技術の変遷; 柿谷均, 生物工学会誌,
Vol.87, No.11, p548-549 (2009).
- 化学的に見たdopamine,およびそのアゴニスト,アンタゴニストと受容体の相互作用;
諸岡良彦, 平井憲次, 清水高子, 臨床精神薬理,
Vol.12, No.11, p2353-2371 (2009).
- Synthesis of novel ageladine A analogs showing more
potent matrix metalloproteinase (MMP)-12 inhibitory
activity than the natural product; N. Ando and S.
Terashima, Bioorganic & Medicinal Chemistry
Letters, Vol.19, No.18, p5461-5463 (2009).
- Synthesis and Biological Activity of Enantiomeric Pairs
of 5-(Alk-2-enyl)thiolactomycin and 5-[(E)-Cycloalk-2-enylidenemethyl]thiolactomycin
Congeners; K. Ohata and S. Terashima, Chemical &
Pharmaceutical Bulletin, Vol.57, No.9, p920-936
(2009).
- Cp2Ni-KOt-Bu-BEt3 (or PPh3)
Catalyst System for Direct C-H Arylation of Benzene,
Naphthalene, and Pyridine; O. Kobayashi, D. Uraguchi and
T. Yamakawa, Organic Letters, Vo.11, No.12, p2679?2682
(2009).
- Synthesis of α-trifluoromethylstyrene derivatives via
Ni-catalyzed cross-coupling of
2-bromo-3,3,3-trifluoropropene and aryl Grignard
reagents; O. Kobayashi, D. Uraguchi, T. Yamakawa, Journal
of Fluorine Chemistry, Vol,130, No.6, p591-594
(2009).
- Nickel-Catalyzed Vinylation of Aryl Chlorides and
Bromides with Vinyl ZnBr·MgBrCl; T. Yamamoto and
T. Yamakawa, Journal of Organic Chemistry, Vol.74,
No.9, p3603?3605 (2009).
- Synthesis of α-trifluoromethylstyrene derivatives via
Pd-catalyzed cross-coupling of
2-bromo-3,3,3-trifluoropropene and arylmagnesium
bromides; O. Kobayashi, D. Uraguchi and T. Yamakawa, Journal
of Molecular Catalysis A: Chemical, Vol.302, No.1-2,
p7-10 (2009).
- Synthesis and Properties of Silicon-containing Polymers
Having Cyclic Silphenylenesiloxane Moieties; K. Noguchi,
E. Akiyama, H. Ito, Y. Nagase, Transaction of the
Materials Research Society of Japan, Vol.34, No.2,
p351-354 (2009).
- Efficient synthesis and biological activity of
enantiomeric pairs of thiolactomycin and its 3-demethyl
derivative;K. Ohata and S. Terashima, Tetrahedron,
Vol.65, No. 11, p2244-2253 (2009).
- 不斉水素化反応の安価な新規触媒系の開発;小林
修, 触媒, Vo.50, No.4, p371 (2008).
- Catalytic trifluoromethylation of uracil to
5-trifluoromethyluracil by use of CF3I and its
industrial applications;D. Uraguchi, K. Yamamoto, Y.
Ohtsuka, K. Tokuhisa, T. Yamakawa, Applied Catalysis
A: General, Vol.342, p137-143 (2008).
- Comparative study on syntheses of
1,3,5-trimethoxy-1,3,5-triisopropyl- cyclotrisiloxane;M.
Ochiai, E. Akiyama, T. Ueno, K. Kawano, T. Hayakawa, N.
Oshima, Silicon Chemistry, Vol.3, No.6, p307-312
(2008).
- Synthesis and biological activity of enantiomeric
pairs of 5-[(E)-cycloalk-
2-enylidenemethyl]thiolactomycin congeners;K. Ohata and
S. Terashima, Bioorganic & Medicinal Chemistry
Letters, Vol.18, No.20, p5598-5600 (2008).
- Cross-Coupling Reaction of Oxazoles; M. Inoue, Mini-Reviews
in Organic Chemistry, Vol.5, No.2, p77-84 (2008).
- パラジウム触媒を用いたアリールアミン類と2-ブロモ-3,3,3-トリフルオロプロペンとのカップリング反応;木野達人、長瀬
裕、堀野良和、山川 哲, 東海大学紀要工学部,
Vol.47, No.2, p15-24 (2007).
- Pd-catalyzed coupling of arylamines and
2-bromo-3,3,3-trifluoropropene;T. Kino, Y. Nagase, Y.
Horino, T. Yamakawa, Journal of Molecular Catalysis A:
Chemical 282, p34?51(2008).
- 仮想スクリーニングによる新規4-ヒドロキシフェニルピルビン酸ジオキシゲナーゼ(4-HPPD)阻害剤の探索;柿谷均、平井憲次、佐藤幸治,
玉川大学学術研究所紀要, p19-24 (2007).
- Enantioselective Total Synthesis of (+)-Ottelione A,
(-)-Ottelione B, (+)-3-epi-Ottelione A and
Preliminary Evaluation of Their Antitumor Activity;0.H.
Araki, M. Inoue, T. Suzuki, T. Yamori, M. Kohno, K.
Watanabe, H. Abe, T. Katoh, Chemistry A European
Journal 13, p9866-9881 (2007).
- マイクロリアクター;山川哲, 環境化学の事典,
p342-343 (2007).
- Synthesis of Poly [(tetraphenyl-p-silphenylenesiloxane)-co-(tetra-methyl-p-
silphenylenesiloxane)]s and the Physical Properties of
Their Films;H. Ito, E. Akiyama, Y. Nagase, and S.
Fukui, Polymer Journal, Vol.39, No.5, p471-477
(2007).
- Enhanced heterologous production of eicosapentaenoic acid
in Escherichia coli cells that co-express
eicosapentaenoic acid biosynthesis pfa genes and
foreign DNA fragments including a high-performance
catalase gene, vktA;Y. Orikasa, Y. Ito, T.
Nishida, K. Watanabe, N. Morita, T. Ohwada, I. Yumoto, H.
Okuyama, Biotechnology Letters 29, p803-809
(2007).
- Iterative two-step strategy for C2-C4' linked
poly-oxazole synthesis using Suzuki-Miyaura
cross-coupling reaction;H. Araki, T. Katoh and M.
Inoue, Tetrahedron Letters 48, p3713-3717 (2007).
- 除草活性を有する新規イミダゾール-4-カルボキサミド誘導体の合成研究;若松晋平、内田淳、横田和加子、平井憲次、長瀬裕,
東海大学紀要工学部, Vol.47, No.1, p5-14
(2007).
- Synthesis and matrix metalloproteinase(MMP)-12 inhibitory
activity of ageladine A and its analogs; N. Ando and S.
Terashima, Bioorganic & Medicinal Chemistry
Letters 17, p4495-4499 (2007).
- Synthesis and biological activity of enantiomeric pairs
of 5-vinylthiolactomycin congeners;K. Ohata and S.
Terashima, Bioorganic & Medicinal Chemistry
Letters 17, p4070-4074 (2007).
- 中性スフィンゴミエリナーゼ阻害剤(+)-スキホスタチンの全合成;井上宗宣、横田和加子、加藤正,
有機合成化学協会誌, Vol.65, No.4,
p358-369 (2007).
- Enantioselective Total Synthesis of (+)-Scyphostatin, a
Potent and Specific Inhibitor of Neutral Sphingomyelinase;M.
Inoue, W. Yokota, T. Katoh, Synthesis 2007,
p622-637 (2007).
- Bacterial Genes Responsible for the Biosynthesis of
Eicosapentaenoic and Docosahexaenoic Acids and Their
Heterologous Expression;H. Okuyama, Y. Orikasa, T.
Nishida, K. Watanabe, and N. Morita, Applied and
Environmental Microbiology, Vol.73, No.3, p665-670
(2007).
- Ambipolar Carrier Transport in Amorphous
Bis(triazinyl)arenes and Their Application in OLED; H.
Aihara, N. Yanai, T. Yamakawa, T. Tanaka* and M. Sato, Transactions
of the Materials Research Society of Japan, 32(2),
p333-336 (2006).
- The domain structure and functional compatibility of the
phospho- pantetheinyl transferases responsible for the
biosynthesis of n-3 long-chain polyunsaturated
fatty acids;Y. Orikasa, T. Nishida, K. Watanabe, N.
Morita, and H. Okuyama, Current Advances in the
Biochemistry and Cell Biology of Plant Lipids:
Proceedings of the 17th International Symposium on Plant
Lipids (ISPL), p169-173 (2006).
- Evaluation of the antioxidative effects of
eicosapentaenoic acid by growth inhibition testing on
plates using Escherichia coli transformed with pfa
genes;T. Nishida, Y. Orikasa, K. Watanabe, N. Morita
and H. Okuyama, urrent Advances in the Biochemistry
and Cell Biology of Plant Lipids: Proceedings of the 17th
International Symposium on Plant Lipids (ISPL), p116-119
(2006).
- A Novel MO Precursor for Metal Tantalum and Tantalum
Nitride Film;K. Sekimoto, T. Furukawa, N. Oshima, K.
Tada, and T. Yamakawa, Materials Research Society
Symposium Proceedings, Vol.914, p161-166 (2006).
-
パラジウム―セピオライト触媒による有機合成反応;森嘉彦,山川哲,
東ソー研究・技術報告, Vol.50, p23-30
(2006).
- 1,3,5-トリアジン化合物の合成と電子輸送性;田中剛,望月修,佐藤優,相原秀典,山川哲,
東ソー研究・技術報告, Vol.50, p9-14 (2006).
- Preparation of Fully Aromatic Polysilarylenesiloxanes by
Melt Polycondensation and Their Thermal Properties;H.
Ito, E. Akiyama, Y. Nagase, A. Yamamoto and S. Fukui, Polymer
Journal, Vol.38, No.10 p1068-1073 (2006).
- Thermal and Physical Properties of
Poly(tetraphenyl-p-silphenylene-siloxane
-co-tetramethyl-p-silphenylenesiloxanes);H. Ito, E.
Akiyama, Y. Nagase and S. Fukui, Transactions of the
Materials Research Society of Japan 31, No.4,
p1065-1068 (2006).
- The cell membrane-shielding function of eicosapentaenoic
acid for Escherichia coli against exogenously
added hydrogen peroxide;T. Nishida, Y. Orikasa, K.
Watanabe, H. Okuyama, FEBS Letters 580, p6690-6694
(2006).
- Synthetic Studies toward GKK1032s, Novel Antibiotec
Antitumor Agents: Enantioselective Synthesis of the Fully
Elaborated Tricyclic Core via an Intramolecular
Diels-Alder Cycloaddition;M. Asano, M. Inoue, K.
Watanabe, H. Abe, and T. Katoh, The Journal of Organic
Chemistry, Vol.71, NO.18, p6942-6951(2006).
- Recombinant production of docosahexaenoic acid in a
polyketide biosynthesis Mode in Escherichia coli;Y.
Orikasa, T. Nishida, A. Yamada, R. Yu, K. Watanabe, A.
Hase, N. Morita, and H. Okuyama, Biotechnology Letters
28, p1841-1847 (2006).
- A phosphopantetheinyl transferase gene essential for
biosynthesis of n?3 polyunsaturated fatty acids from Moritella
marina strain MP-1;Y. Orikasa, T. Nishida, A. Hase,
K. Watanabe, N. Morita, and H. Okuyama, FEBS Letters
580, p4423?4429 (2006).
- Escherichia coli engineered to produce
eicosapentaenoic acid becomes resistant against oxidative
damages;T. Nishida, Y. Orikasa, Y. Itoh, R. Yu, A.
Yamada, K. Watanabe, H. Okuyama, FEBS Letters 580,
p2731-2735 (2006).
- A Novel Synthesis of the 2-Aminoimidazol-4-carbaldehyde
Derivatives, Versatile Synthetic Intermediates for
2-Aminoimidazole Alkaloids;N. Ando and S. Terashima, Synlett,
No.17, p2836-2840 (2006).
- Convergent and enantioselective total synthesis of
(-)-nalanthalide, a potential Kv1.3 blocking
immunosuppressant;T. Abe, K. Iwasaki, M. Inoue, T.
Suzuki, K. Watanabe and T. Katoh, Tetrahedron Letters
47, p3251-3255 (2006).
- Efficient synthesis of enantiomeric pairs of
thiolactomycin and its 3-demethyl derivative;K. Ohata
and S. Terashima, Tetrahedron Letters 47,
p2787-2791 (2006).
-
全芳香族ポリシルアリーレンシロキサンの合成と熱物性および耐熱性機能材料への展開;伊藤仁士,秋山映一,長瀬裕,
高分子加工, 55巻5号, p19-26 (2006).
- An industrially usable Pd-catalyzed carboalkoxylation of
1,2-dibromo -3,3,3-trifluoropropane to tert-butyl
trifluoromethacrylate in the presence of an inorganic
base, Y. Horino, N. Wakasa, T. Fuchikami and T. Yamakawa,
Journal of Molecular Catalysis A: Chemical,
Vol.258, No.1-2, p152-158 (2006).
- Enantiocontrolled synthesis of the epoxycyclohexenone
moieties of scyphostatin, a potent and specific inhibitor
of neutral sphingomyelinase; T. Katoh, T. Izuhara, W.
Yokota, M. Inoue, K. Watanabe, A. Nobeyama, T. Suzuki and
Tetrahedron, Vol.62, No.7, p1590-1608 (2006).
- Synthesis and Reaction of the First Oxazol-4-ylboronates:
Useful Reagents for the Preparation of the
Oxazole-Containing Biaryl Compounds, H. Araki, T. Katoh,
M. Inoue, Synlett, No.4, p555-558 (2006).
- Synthesis and Thermal Properties of Fully Aromatic
Polysilarylenesiloxanes; H. Ito, E. Akiyama, Y. Nagase,
A. Yamamoto, S. Fukui, Polymer Journal, Vol.38,
No.2 p109-116 (2006)
- 新規1,2,4-トリアジン誘導体の合成と生物活性;内田淳,大野竜太,鹿倉光一,矢野智行,鵜飼貞行,山田修,佐藤幸治,平井憲次,玉川大学学術研究所紀要,第11号,p11-19
(2005).
- 酵素トルエンモノオキシゲナーゼを利用した選択的酸化反応技術の開発;
飯田寛, 丸山高廣, 小林秀峰, 柿谷均, 東ソー研究・技術報告,
第49巻 別冊, p3-13 (2005).
- 平成17年度論文賞対象論文の概要とその研究背景;
柿谷均, 日本農薬学会誌, Vol.30, No.3,
p246-248 (2005).
- 除草剤ペントキサゾンの開発; 平井憲次, 堀正大,
ファインケミカル, 2005年7月, Vol.34,
No.7, p49-56 (2005).
- Enantioselective Total Synthesis of (-)-Candelalide A, a
Novel Blocker of the Voltage-Gated Potassium Channel
Kv1.3 for an Immunosuppresive Agent; K. Watanabe, K.
Iwasaki, T. Abe, M. Inoue, K. Ohkubo, T. Suzuki, and T.
Katoh, Organic Letters, Vo.7, No.17, p3745-3748
(2005).
- Model Studies towards the Total Synthesis of GKK1032s,
Novel Antibiotic Anti-Tumor Agents: Enantioselective
Synthesis of the Alkyl Aryl Ether Portion of GKK1032s; M.
Asano, M. Inoue, T. Katoh, SYNLETT, No.17,
p2599-2602 (2005).
- Enantioselective Synthesis of the Tricyclic Core of
GKK1032, Novel Antibiotic Anti-Tumor Agents, by Employing
an Intramolecular Diels-Alder Cycloaddition Strategy; M.
Asano, M. Inoue, T. Katoh, SYNLETT, No.10,
p1539-1542 (2005).
- 構造ゲノム科学の進展とその応用; 柿谷均,
技術士, 平成17年3月号, p12-15 (2005)
- Total Synthesis of (+)-Scyphostatin, a Potent and
Specific Inhibitor of Neutral Sphingomyelinase; M. Inoue,
W. Yokota, M. G. Murugesh, T. Izuhara, and T. Katoh,
Angewandte Chemie International Edition, 43,
p4207-4209 (2004)
- A Novel Iridium Precursor for MOCVD; 河野和久,
高森真由美, 多田賢一, 山川哲, 大島憲昭,
亘理総一, 藤沢浩訓, 清水勝, 東ソー研究・技術報告,
第48巻, p2-8 (2004)
- A Novel Iridium Precursor for MOCVD; K. Kawano M.
Takamori, T. Yamakawa, S. Watari, H. Fujisawa, M.
Shimizu, H. Niu, and K. Ohshima, Materials Research
Society Symposium Proceedings, Vol.784, p145-150
(2004)
- Characterization of the Eicosapentaenoic Acid
Biosynthesis Gene Cluster from Shewanella sp. Strain
SCRC-2738; Y. Orikasa, A. Yamada, R. Yu, Y. Ito, T.
Nishida, I. Yumoto, K.Watanabe, and H. Okuyama, Cellular
and Molecular Biology, 50 (5), p625-630 (2004)
- Synthesis and Herbicidal Activity of New
1-Alkyl-3-aryloxypyrazole-4-carboxamide Derivatives; R.
Ohno, A. Watanabe, M. Nagaoka, T. Ueda, H. Sakurai, M.
Hori, and K. Hirai, Journal of Pesticide Science,
Vol.29, No.2, p96-104 (2004)
- Alkylation of
Ethylenediamine with Alcohols by Use of Cu-based
Catalysts in the Liquid Phase; T. Yamakawa, I. Tsuchiya,
D. Mitsuzuka, and T. Ogawa, Catalysis Communications,
5, p291-295 (2004)
- Whole-Body β-Oxidation of Docosahexaenoic Acid Is
Decreased under n-3 Polyunsaturated Fatty Acid
Insufficiency as Assessed by a 13CO2
Breath Test Using [U-13C] Fatty Acids; H.
Waki, K. Watanabe, H. Ishii, Y. Tanaka, S. Shumiya and S.
Ando, Journal of Oleo Science, Vol. 53 No.3,
p135-142 (2004)
- Synthesis and Herbicidal Activity of New
Pyrazole-4-carboxamide Derivatives; R. Ohno, A. Watanabe,
T. Matsukawa, T. Ueda, H. Sakurai, M. Hori and K. Hirai, Journal
of Pesticide Science 29, p15-26 (2004).
- 破線状ガイドライン構造のチャンネルをもつマイクロリアクタによる水と有機溶媒の分離;
山川哲、押手浩之、片山晃治、二見達、大川朋裕、西沢恵一郎,
化学工学論文集 30巻1号, p95-97 (2004).
- Three-Dimensional Modeling of Plant
4-Hydroxyphenylpyruvate Dioxygenase, a Molecular Target
of Triketone-Type Herbicides; H. Kakidani and K. Hirai, Journal
of Pesticide Science 28, p409-415 (2003).
- Enantioselective Total Synthesis of 3-epi-Ottelione A;
H. Araki, M. Inoue and T. Kato, SYNLETT, No.15,
p2401-2043 (2003).
- Synthetic Studies of Kampanols, Novel p21ras
Farnesyltransferase Inhibitors : an Efficient Synthesis
of the Tetracyclic ABCD Ring System of Kampanols; K.
Iwasaki, M. Nakatani, M. Inoue and T. Katoh, Tetrahedron
59, p8763-8773 (2003).
- Total Synthesis and Absolute Configuration of Otteliones
A and B, Novel and Potent Antitumor Agents from a
Freshwater Plant; H. Araki, M. Inoue and T. Katoh, Organic
Letters vol.5 no.21, p3903-3906 (2003).
- Enantioselective Total Synthesis of (+)-Aureol via a
BF3・Et2O-promoted Rearrangement/ Cyclization
Reaction of (+)-Arenarol; M. Nakatani, M. Nakamura, A.
Suzuki, T. Fuchikami, M. Inoue and T. Katoh, Arkivoc
Part (xiii), p45-57 (2003).
- 除草剤・植物成長調節剤の動向;
平井憲次、大野竜太, CMC出版 「新農薬開発の最前線」,
p135-189 (2003).
- Novel efficient synthesis of an enantiomeric pair of
tricycloillicinone; S. Furuya and S. Terashima, Tetrahedron
Letters 44, p6875-6878 (2003).
- Synthetic Studies of Cazinophilin. Part 4; Chemical and
Biological Properties of Carzinophilin Analogues; M.
Hashimoto, M. Matsumoto, K. Yamada and S. Terashima, Tetrahedron
59, p3089-3097 (2003).
- Synthetic Studies of Carzinophilin. Part 3: Synthetic
Approach toward Carzinophilin and Successful Synthesis of
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- Synthetic Studies of Carzinophilin. Part 2: Synthesis of
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- Synthetic Studies of Carzinophilin. Part 1: Synthesis of
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- Synthetic Studies on Himbacine, a Potent Antagonist of
the Muscarinic M2 Subtype Receptor.
Part 2: Synthesis and Muscarinic M2 Subtype Antagonistic
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C-3 Position of Lactone Moiety
M. Takadoi, K. Yamaguthi and S. Terashima, Bioorganic
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A. Suzuki, M. Nakatani, M. Nakamura, K. Kawaguchi, M.
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T. Katoh and S. Terashima, Latest Frontiers of organic
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- A New Strategy toward the Total Synthesis of Stachyflin,
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M. Takadoi, K. Yamaguchi** and S. Terashima, Bioorganic
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- Synthesis and Muscarinic M2 Subtype Antagonistic Activity
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M. Takadoi, S. Terashima, Bioorganic and Medicinal
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- Model studies toward scyphostatin:synthesis of
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Y. Fukuda, S. Seto, H. Furuta, H. Ebisu, Y. Oomori, S.
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- Liquid crystalline coumarin polymers. II: Photo-chemistry
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- Enantiocontrolled synthesis of
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- A Novel Synthesis of Avermectin B1a From Avermectin B2a
T.Katoh, E.Itoh, S.Terashima, Heterocycles,
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antagonist of the galanin receptor subtype GalR1:
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- Novel polyamides for second-order nonlinear optics with
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- Palladium diaqua and hydroxo complexes with
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- A heterozygous mutation of β-actin associated with
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Y.Wu, Q.Zhang, A.Kanazawa, T.Shiono, T.Ikeda, Y.Nagase , Macromolecules,
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M.Takadoi, T.Katoh, A.Ishiwata, S.Terashima, Tetrahedron
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- Selection of cDNAs encoding putative type II membrane
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- Transition Metal-catalyzed Dehydrogenative Silylation of
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- Stereospecific Nucleophilic Substitution of Optically
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- Biological Activities of 1,1,6-Trisubstituted Indanes:
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- A new class of second-order non-linear optical material:
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- Synthetic Studies of Huperzine A and Its Fluorinated
Analogues.2. Synthesis and Acetylcholinesterase
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- Synthetic Studies of Huperzine A and Its Fluorinated
Analogues.1. Novel Asymmetric Syntheses of an
Enantiomeric Pair of Huperzine A
S.Kaneko, T.Yoshino, T.Katoh, S.Terashima, Tetrahedron,
Vol.54, No.21, 5471(1998).
- Identification and Characterization of a Novel SH3-Domain
Binding Protein, Sab, Which Preferentially Associates
with Bruton's Tyrosine Kinase(Btk)
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- Photochemical Phase-Transition Behavior of Polymer Liquid
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- Structure-Activity Relationship of Norzoanthamine
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- Practical Synthesis of
(2S,3S)-3-Amino-2-hydroxy-4-phenylbutyric Acid, A Key
Component of HIV Protease Inhibitors
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- Enantioselective Addition of Enol Silyl Ethers to Imines
Catalyzed by Palladium Complexes; A Novel Way to
Optically Active Acylalanine Derivatives
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- (4R,5S)-4,5-DIPHENYL-3-VINYL-2-OXAZOLIDINONE
T. Akiba, O. Tamura, S. Terashima, Organic Synthesis,
Vol.75(1997).
- Structually Simplified Zaragozic Acid
(Squalestatin):Stereoselective Preparation of a
3,4-Unsubstituted Derivative
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- Stereo-and Regioselective Bromination of
1,5-Cyclooctadiene Derivatives and Their Substitution
Reactions with Organocopper Reagents
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- Polymeric percutaneous drug penetration enhancer
Synthesis and enchancing property of PEG/PDMS block
copolymer with a cationic end group
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of Controlled Release, 49, 229(1997).
- Special Folding Pathway to Tetramer Only through the
Micelle State of the Corticotropin-Releasing Factor
H. Morii, H. Uedaira, M. Ishimura, S. Kidokoro, T.
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No.49,15538(1997).
- Studies on Synthesis of γ-Butyrolactone by the
Hydrogenation of Maleic Anhydride and Its Derivatives.
The Catalytic Properties of Ruthenium Complex Catalysts
and the Effect of Additives
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Technology(中国), Vol.26, No.7, 425(1997).
- Effect of Siloxane Spacer on Photochemical Phase
Transition Behavior of Polymer Liquid Crystals with
Azobenzene Moieties in the Side Chain
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- Absolute Configuration of Norzoanthamine, a Promising
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- A Stereoselective Synthesis of
4-O-Methyl-13-Desacetyl-12,13-Di-O-Benzylcarzinophilin
M. Hashimoto, S. Terashima, Heterocycles, Vol.47,
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- Norzoanthamine Suppresses PTH Stimulated IL-6 Production
inVitro and Bone Resorption in Vivo
T. Tsuji, K. Yamaguchi, M. Yada, K. Yamada, D. Uemura,
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- An Enantioselective Synthesis of Natural (-)-Huperzine a
Via Cinchona Alkaloids-Promoted Asymmetric Michael
Reaction
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Vol.46, 27(1997).
- Development of Chemical Substances Regulating Biofilm
Formation
A. Yamada, H. Kitamura, K. Yamaguchi, S. Fukuzawa, C.
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- Novel Syntheses of Optically Active CC-1065,
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- Total Synthesis of Antitumor Antibiotic FR900482
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- Suppression of Colon Carcinogenesis by Docosahexaenoic
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- Structure-Activity Relationship of Cantharidin
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- Antibacterial Activity of (+/-)
6-Benzyl-1-(3-carboxypropyl)indane; A Possible Way to
IdentifyLeading Novel Anti-H. pylori Agents
N. Numao, Y. Hirota, A. Iwahori, M. Sasatsu, I. Kondo, K.
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- Novel concept for non-destructive readout method for
photochromic rewriteable memory devices
J. Abe, N. Nemoto, Y. Nagase, Y. Shirai, Chemical
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- Studies Toward the Synthesis of Popolohuanone E :
Synthesis of Natural(+)-Arenarol Related to the Proposed
Biogenetic Precursor of Popolohuanone E
H. Kawano, M. Itoh, T. Katoh, S. Terashima, Tetrahedron
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- A new synthetic approach to side-chain liquid crystalline
polyacrylates containing siloxane spacers and their
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- Lipid and Fatty Acid Compositions of a Novel
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K. Watanabe, C. Ishikawa, I. Ohtsuka, M. Kamata, M.
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- A Novel Synthesis of (+)-Duocarmycin SA
Y. Fukuda, S. Terashima, Tetrahedron Lett.,
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- Novel Thermotropic Liquid Crystals without a Rigid Core
Formed by Amphiphiles Having Phosphonium Ions
A. Kanazawa, O. Tsutsumi, T. Ikeda, Y. Nagase, J. Am.
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- Human cDNA Encoding a Novel TGF-βSuperfamily Protein
Highly Expressed in Placenta
M. Yokoyama-Kobayashi, M. Saeki, S. Sekine, S. Kato, J.
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- Lewis Base Catalyzed Trifluoromethylation of Carbonyl
Compounds with Trialkyl(trifluoromethyl)silanes
T. Hagiwara, T. Kobayashi, T. Fuchikami, Main Group
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- Manipulation of Dipole Moment and Hyperpolarizability
Based on Heterocyclic Pyridinium Betaine Structures:Ab
Initio and INDO MO Calculations
J. Abe, Y. Shirai, N. Nemoto, Y. Nagase, J. Phys.
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- Time course of bone biomechanical parameters in
ovariectomized mice
K. Yamaguchi, T. Hayama, T. Makita, T. Tsuji, J. Bone
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- Fatty Acid Synthesis of an Eicosapentaenoic
Acid-Producing Bacterium: De Novo Synthesis,
ChainElongation, and Desaturation Systems
K. Watanabe, K. Yazawa, K. Kondo, A. Kawaguchi, J.
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- Synthesis of
2-O-(3-O-Carbamoyl-?-D-mannopyranosyl)-L-gulopyranose:
Sugar Moiety of Antitumor Antibiotic Bleomycin
T. Oshitari, M. Shibasaki, T. Yoshizawa, M. Tomita, K.
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- Total Synthesis of an Enantiomeric Pairof FR900482. 3.
Completion of the Synthesis by Assembling the Two
Segments
T. Katoh, Y. Nagata, T. Yoshino, S. Nakatani, S.
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10253(1997).
- A new class of second-order non-linear optical material:
stilbazolium benzimidazolate covalently bound to polymer
backbone
N. Nemoto, J. Abe, F. Miyata, Y. Shirai, Y.Nagase, J.
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- Total Synthesis of an Enantiomeric Pair of FR900482. 2.
Syntheses of the Aromatic and the Optically Active
Aliphatic Segments
T. Yoshino, Y. Nagata, E. Itoh, M. Hashimoto, T. Katoh,
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- Total Synthesis of an Enantiomeric Pair of FR900482. 1.
Synthetic and End-Game Strategies
T. Katoh, E. Itoh, T. Yoshino, S. Terashima, Tetrahedron,
Vol.53, No.30, 10229(1997).
- Photochemical phase transition behaviour of polymer
azobenzene liquid crystals with flexible siloxane units
as a side-chain spacer
A. Kanazawa, S.Hirano, A. Shishido, M. Hasegawa, O.
Tsutsumi, T. Shiono, T. Ikeda, Y. Nagase, E. Akiyama, Y.
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293(1997).
- 1,2-Bis(dimethylphenylsilyl)tetrafluoroethane.
Application to the Trifluorovinylation and
Tetrafluoroethylenation of Carbonyl Compounds
T. Hagiwara, T. Fuchikami, Chem. Lett., No.8,
787(1997).
- Unique Reactivity of Aminoketones in the
Trifluoromethylation with
Trialkyl(trifluoromethyl)silanes
T. Hagiwara, H. Mochizuki, T. Fuchikami, Synlett,
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- DHAの生化学
M. Shikano, K. Yazawa, Asthma, Vol.10, No.3,
39(1997).
- On the Antibacterial Activity of Normal and Reversed
Magainin 2 Analogs against Helicobacter pylori
A. Iwahori, Y. Hirota, R. Sampe, S. Miyano, N. Takahashi,
M. Sasatsu, I. Kondo, N. Numao, Biol. Pharm. Bull.,
Vol.20, No.7, 805(1997).
- Antibacterial Activity of Two Alkylamines Integrated an
Indane Scaffold: Mimicry of a Complementary Unit on +Magainin
2
N. Numao, A. Iwahori, Y. Hirota, M. Sasatsu, I. Kondo, K.
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- Synthesis and Antitumor Activity of Novel
Cyclopropapyrroloindole(CPI) Derivatives Bearing
Methoxycarbonyl and Trifluoromethyl Groups
Y. Fukuda, H. Furuta, F. Shiga, Y. Oomori, Y. Kusama, H.
Ebisu, S. Terashima, Bioorg. Med. Chem. Lett.,
Vol.7, No.13, 1683(1997).
- Stable Diaqua Palladium(U)Complexes of BINAP and
Tol-BINAP as Highly Efficient Catalysts for Asymmetric
Aldol Reactions
M. Sodeoka, R. Tokunoh, F. Miyazaki, E. Hagiwara, M.
Shibasaki, Synlett, No.5, 463(1997).
- Synthesis and Lewis Acid-Catalyzed Nucleophilic
Substitution of Chiral 1-Alkoxyalkyl Carboxylates
H. Matsutani, S. Ichikawa, J. Yaruva, T. Kusumoto, T.
Hiyama, J. Am. Chem. Soc., Vol.119, No.19,
4541(1997).
- Synthesis of (+/-)-12-Fluorohuperzine A, a Novel
Acetylcholinesterase Inhibitor
S. Kaneko, M. Shikano, T. Katoh, S. Terashima. Synlett,
No.5, 447(1997) .
- HSDJ, a Human Homolog of DnaJ, Is Farnesylated and Is
Involved in Protein Import into Mitochondria
M. Kanazawa, K. Terada, S. Kato, M. Mori. J. Biochem.,
Vol.121, No.5, 890(1997).
- N-(Carbamoylmethyl)pyridinium Perchlorate and
N-(Carbamoylmethyl)-N'-methyl-4,4'-bipyridinium
Diperchlorate Hydrate
K. Sakai, Y. Ikuta, M. Shiomi, T. Tamane, Y. Tomita, T.
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331(1997).
- Heterocyclic Pyridinium Betaines, A New Class of
Second-Order Nonlinear Optical Materials: Combined
Theoretical and Experimental Investigation of First-Order
Hyperpolarizability through ab Initio, INDO , and
Hyper-Rayleigh Scattering
J. Abe, Y. Shirai, N. Nemoto, F. Miyata, Y. Nagase, J.
Phys. Chem. B, Vol.101, No.4, 576(1997).
- 二量体型液晶化合物の構造と物性
T. Kusumoto, T. Hiyama, 染料と薬品, Vol.42, No.4,
85(1997).
- S. Kaneko, T. Yoshino, T. Katoh, S. Terashima, Tetrahedron:
Asymmetry, Vol.8, No.6, 829(1997).
A novel enantioselective synthesis of the key
intermediate of (-)-huperzine A employing asymmetric
palladium-catalyzed bicycloannulation
- 「生命論」を生物物理から発信しよう
A. Wada, 生物物理, Vol.37, No.2, 85(1997).
- An Expeditious Synthesis of
(2R,3S)-3-tert-Butoxycarbonylamino-1-isobutylamino-4-phenyl-2-butanol,
a Key Building Block of HIV Protease Inhibitors
N. Shibata, T. Katoh, S. Terashima, Tetrahedron Lett.,
Vol.38, No.4, 619(1997).
- Synthesis and Antitumor Activity of Novel
Cyclopropapyrroloindole (CPI)Derivatives Bearing
Bis(Methoxycarbonyl)Groups
Y, Fukuda, Y. Oomori, Y. Kusama, S. Terashima, Bioorganic
Med. Chem. Lett., Vol.7, No.6, 749(1997).
- Evaluation of Skin Permeability of Drugs by Newly
Prepared Polymer Membranes
Y. Yamaguchi, T. Usami, H. Natsume, T. Aoyagi, Y. Nagase,
K. Sugibayashi, Y. Morimoto, Chem. Pharm. Bull.,
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- Synthesis of Reversed Magainin 2 Analogs Enhanced
Antibacterial Activity
A. Iwahori, Y. Hirota, R. Sampe, S. Miyano, N. Numao, Biol.
Pharm. Bull., Vol.20, No.3, 267(1997).
- 縮合系ポリマーからなる非線形光学材料
N. Nemoto, 高分子, Vol.46, No.3, 132(1997)
- Theoretical Study of Hyperpolarizabilities of Spirolinked
Push-Pull Polyenes
J. Abe, Y. Shirai, N. Nemoto, Y. Nagase, J. Phys.
Chem. A, Vol.101, No.1, 1(1997).
- Theoretical Study of the Third-Order Nonlinear Optical
Properties of Spiro-Linked Polyene
J. Abe, Y. Shirai, N. Nemoto, Y. Nagase, T. Iyoda, J.
Phys. Chem. B, Vol.101, No.2, 145(1997).
- Polyamides for Nonlinear Optics: Side-Chain All
Donor-Attached NLO-phores versus Side-Chain Alternating
Donor-Attached and Acceptor-Attached NLO-phores
N. Nemoto, F. Miyata, Y. Nagase, J. Abe, M. Hasegawa, Y.
Shirai, Chem. Mater., Vol.9, No.1, 304(1997).